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3-Methyl-GABA

  Cat. No.:  DC40224  
Chemical Structure
1216629-00-3
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More than 5000 active chemicals with high quality for research!
Field of application
3-Methyl-GABA is an activator of GABA aminotransferase with anticonvulsant activity.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 1216629-00-3
Chemical Name: 3-Methyl-GABA
SMILES: O=S(C1=C2C=CC=C(S(=O)(O)=O)C2=CC=C1)(O)=O.O=C(O)CC(C)CN.O=C(O)CC(C)CN
Formula: C20H30N2O10S2
M.Wt: 522.59
Sotrage: Please store the product under the recommended conditions in the Certificate of Analysis.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
Cat. No. Product name Field of application
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DC46487 LU-32-176B LU-32-176B, a GABA transporter 1(GAT1) selective inhibitor, is found to exert a synergistic anticonvulsant action with GAT2 transport inhibitor EF1502. LU-32-176B inhibits neurons, astrocytes and mGAT1 with the IC50 values of 2μM, 1μM, 4μM, respectively.
DC46367 Lesogaberan hydrochloride Lesogaberan (hydrochloride) is a potent and selective GABAB receptor agonist with an EC50 of 8.6 nM for human recombinant GABAB receptors. Binding affinity (Kis) of 5.1 nM and 1.4 μM for rat brain GABAB and GABAA receptors, respectively.
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