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680C91

  Cat. No.:  DC48330   Featured
Chemical Structure
163239-22-3
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More than 5000 active chemicals with high quality for research!
Field of application
680C91 is an orally active, selective tryptophan 2,3-dioxygenase (TDO) inhibitor with a Ki of 51 nM. TDO is the key enzyme of tryptophan catabolism. 680C91 can be used for the research of cancer immunotherapy and Alzheimer’s Disease.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 163239-22-3
Chemical Name: 680C91
Synonyms: 1H-Indole,6-fluoro-3-[(1E)-2-(3-pyridinyl)ethenyl]-;680C91;6-Fluoro-3-[(E)-2-(3-pyridinyl)vinyl]-1H-indole;MC 1443;1H-Indole,6-fluoro-3-[2-(3-pyridinyl)ethenyl]-, (E)-;6-Fluoro-3-[(1E)-2-(3-pyridinyl)ethenyl]-1H-indole
SMILES: FC1C=C2C(C(/C=C/C3=CC=CN=C3)=CN2)=CC=1
Formula: C15H11N2F
M.Wt: 238.25964
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
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