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Apararenone

  Cat. No.:  DC12636   Featured
Chemical Structure
945966-46-1
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More than 5000 active chemicals with high quality for research!
Field of application
Apararenone (MT-3995) is a novel potent, selective non-steroidal mineralocorticoid receptor antagonist for the treatment of diabetic nephropathies and non-alcoholic steatohepatitis..
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 945966-46-1
Chemical Name: N-(4-(4-fluorophenyl)-2,2-dimethyl-3-oxo-3,4-dihydro-2H-benzo[b][1,4]oxazin-7-yl)methanesulfonamide
Synonyms: MT-3995;MT3995
SMILES: CS(NC1C=C2C(=CC=1)N(C1=CC=C(F)C=C1)C(=O)C(C)(C)O2)(=O)=O
Formula: C17H17FN2O4S
M.Wt: 364.391
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: Apararenone (MT-3995) is a novel non-steroidal mineralocorticoid receptor antagonists under development for the treatment of diabetic nephropathies and non-alcoholic steatohepatitis.
In Vivo: Recently, a phase II clinical trial has been initiated among patients with non-alcoholic steatohepatitis (NASH) in Japan[1].
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
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