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NSC 625987

  Cat. No.:  DC20480   Featured
Chemical Structure
141992-47-4
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More than 5000 active chemicals with high quality for research!
Field of application
NSC 625987 is a potent, selective CDK4 inhibitor with IC50 of 0.2 uM, displays >500-fold selectivity over CDK2 (IC50 >100 uM for cdc2/cyclin A, cdk2/cyclin A and cdk2/cyclin E). .
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 141992-47-4
Chemical Name: NSC 625987
Synonyms: 9(10H)-Acridinethione,1,4-dimethoxy-;1,4-dimethoxy-10H-acridine-9-thione;NSC 625987;1,4-DiMethoxy-9(10H)-acridinethione;1,4-Dimethoxy-9-thio(10H)-acridone;Tocris-2152;FT-0711674;HMS3413I05;Q27075829;HY-103380;J-007574;CHEBI:114175;HMS3268N07;CHEMBL1331734;X5RCK1XO4F;Cdk4 Inhibitor II, NSC 625987 - CAS 141992-47-4;UNII-X5RCK1XO4F;SCHEMBL1985563;DTXSID90161912;HMS3229E06;SR-01000597535;MS-23842;141992-47-4;GTPL5951;BRD-K62949423-001-02-3;AKOS022488648;SMP2_000076;NCGC00025358-01;HMS3677I05;CCG-206829;HMS2043P07;CS-0027779;1,4-dimethoxy-9,10-dihydroacridine-9-thione;1,4-Dimethyoxy-9(10H)-acridinone;BDBM59089;NSC-625987;NSC625987;MFCD08276925;NSC 625987, >=97% (HPLC);SR-01000597535-1;NCI60_008225;E98772;Cdk4 inhibitor II;9(10H)-Acridinethione,4-dimethoxy-;1,4-Dimethoxy-9(10H)-acridinethione;1,4-Dimethoxy-9(10H)-acridinethione;9(10H)-Acridinethione, 1,4-dimethoxy-;9(10H)-Acridinethione, 1,4-dimethoxy-;BRD-K62949423-001-03-1;BRD-K62949423-001-03-1;SDCCGSBI-0086742.P003;SDCCGSBI-0086742.P003
SMILES: COC1C2=C(NC3C(C2=S)=CC=CC=3)C(OC)=CC=1
Formula: C15H13NO2S
M.Wt: 271.33422
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: NSC 625987 is a potent, selective CDK4 inhibitor with IC50 of 0.2 uM, displays >500-fold selectivity over CDK2 (IC50 >100 uM for cdc2/cyclin A, cdk2/cyclin A and cdk2/cyclin E).
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
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