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ML 086 (CID-1674999)

  Cat. No.:  DC21317   Featured
Chemical Structure
1177148-36-5
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More than 5000 active chemicals with high quality for research!
Field of application
ML 086 is a potent, specific inhibitor of phosphatase PHOSPHO1 with IC50 of 139 nM, with no activity against TNAP (IC50>100 uM).
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 1177148-36-5
Chemical Name: N,N-dimethyl-3-(3-oxo-1,2-benzothiazol-2-yl)benzamide
Synonyms: ML086;CID-1674999;ML-086;ML 086;CID 1674999;CID1674999
SMILES: C(N(C)C)(=O)C1=CC=CC(N2C(=O)C3=CC=CC=C3S2)=C1
Formula: C16H14N2O2S
M.Wt: 298.36
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: ML 086 is a potent, specific inhibitor of phosphatase PHOSPHO1 with IC50 of 139 nM, with no activity against TNAP (IC50>100 uM); a useful chemical tool to examine the functional role of this enzyme in skeletal mineralization and soft tissue ossification abnormalities.
References: References 1. Stonich D, et al. Probe Reports from the NIH Molecular Libraries Program [Internet]. 2. Bravo Y, et al. Bioorg Med Chem Lett. 2014 Sep 1;24(17):4308-11. View Related Products by Target Protein Phosphatase/PTP
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
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