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RC-3095

  Cat. No.:  DC21560   Featured
Chemical Structure
138147-78-1
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More than 5000 active chemicals with high quality for research!
Field of application
RC-3095 is a gastrin-releasing peptide receptor antagonist, synergizes with gemcitabine to inhibit the growth of human pancreatic cancer CFPAC-1 in vitro and in vivo. RC-3095 inhibit the growth of human glioblastomas in vitro and in vivo. RC3095 inhibits tumor growth and decrease the levels and mRNA expression of epidermal growth factor receptors in H-69 small cell lung carcinoma.R,BRS-1) antagonist.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 138147-78-1
Chemical Name: D-Tpi-Gln-Trp-Ala-Val-Gly-His-Leu-Y(CH2-NH)-Leu-NH2 trifluoroacetate salt
Synonyms: RC 3095;RC3095
SMILES: NC(CC[C@@H](C(N[C@@H](CC1=CNC2=CC=CC=C12)C(N[C@H](C(N[C@H](C(NCC(N[C@H](C(N[C@H](CN[C@H](C(=O)N)CC(C)C)CC(C)C)=O)CC1=CN=CN1)=O)=O)C(C)C)=O)C)=O)=O)NC([C@@H]1NCC2=C(C3=CC=CC=C3N2)C1)=O)=O.FC(C(=O)O)(F)F
Formula: C56H79N15O9.XC2Hf3O2
M.Wt: 1220.34492301941
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: RC-3095 is a bombesin/gastrin releasing peptide receptor antagonist[1].
References: [1]. Konturek SJ, et al. Antagonism of receptors for bombesin, gastrin and cholecystokinin in pancreatic secretion and growth. Digestion. 1991;48(2):89-97.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
2018-0101
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