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MALAT1-IN-1

  Cat. No.:  DC22143   Featured
Chemical Structure
827327-28-6
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More than 5000 active chemicals with high quality for research!
Field of application
MALAT1 inhibitor 5 (Malat1 inhibitor 5) is a selective small molecule targeting of Metastasis-associated lung adenocarcinoma transcript 1 (Malat1/MALAT1 mouse/human), a highly conserved long non-coding RNA; does not affect Neat1 lncRNA levels.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 827327-28-6
Chemical Name: N-(3-methoxybenzyl)-5-(4-methoxyphenyl)-1-methyl-1H-imidazol-2-amine
Synonyms: MALAT1 inhibitor 5|Malat1 inhibitor 5
SMILES: CN1C(C2=CC=C(OC)C=C2)=CN=C1NCC3=CC=CC(OC)=C3
Formula: C19H21N3O2
M.Wt: 323.396
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Publication: 1. Abulwerdi FA, et al. ACS Chem Biol. 2019 Jan 8. doi: 10.1021/acschembio.8b00807.
Description: MALAT1 inhibitor 5 is a potent and specific Malat1 (Metastasis-associated lung adenocarcinoma transcript 1) inhibitor. MALAT1-IN-1 modulated Malat1 downstream genes in a dose-dependent manner without affecting expression of nuclear enriched abundant transcript 1 (Neat1) [1].
References: [1]. Abulwerdi FA, et al. Selective Small-Molecule Targeting of a Triple Helix Encoded by the Long Noncoding RNA, MALAT1. ACS Chem Biol. 2019 Feb 15;14(2):223-235.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
2018-0101
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