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LY2940094

  Cat. No.:  DC22312   Featured
Chemical Structure
1307245-86-8
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More than 5000 active chemicals with high quality for research!
Field of application
LY2940094 is a potent and selective nociceptin receptor antagonist which inhibits excessive feeding behavior in rodents.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 1307245-86-8
Chemical Name: (2-(4-((2-Chloro-4,4-difluoro-spiro(5H-thieno(2,3-C)pyran-7,4'-piperidine)-1'-yl)methyl)-3-methyl-pyrazol-1-yl)-3-pyridyl)methanol
Synonyms: LY2940094;LY 2940094 - Bio-X;4I67US2V8Q;(2-(4-((2'-chloro-4',4'-difluoro-4',5'-dihydrospiro[piperidine-4,7'-thieno[2,3-c]pyran]-1-yl)methyl)-3-methyl-1H-pyrazol-1-yl)pyridin-3-yl)methanol;J3.309.394B;(2-(4-((2-Chloro-4,4-difluoro-spiro(5H-thieno(2,3-C)pyran-7,4'-piperidine)-1'-yl)methyl)-3-methyl-pyrazol-1-yl)-3-pyridyl)methanol;[2-[4-[(2-chloro-4,4-difluorospiro[5H-thieno[2,3-c]pyran-7,4'-piperidine]-1'-yl)methyl]-3-me
SMILES: ClC1=C([H])C2C(C([H])([H])OC3(C=2S1)C([H])([H])C([H])([H])N(C([H])([H])C1=C([H])N(C2=C(C([H])=C([H])C([H])=N2)C([H])([H])O[H])N=C1C([H])([H])[H])C([H])([H])C3([H])[H])(F)F
Formula: C22N4O2F2SclH23
M.Wt: 480.9584
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: LY2940094 is a potent, selective and orally available nociceptin receptor (NOP) antagonist with an Ki of 0.105 nM.
Target: Ki: 0.105 nM (NOP)[1]
References: [1]. Rorick-Kehn LM, et al. A Novel, Orally Bioavailable Nociceptin Receptor Antagonist, LY2940094, Reduces Ethanol Self-Administration and Ethanol Seeking in Animal Models. Alcohol Clin Exp Res. 2016 May;40(5):945-54.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
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