BRD-4592| CAS 2109805-80-1

Cas No.:	2109805-80-1
Chemical Name:	BRD-4592
SMILES:	C1C=CC(C2=CC=C([C@@H]3[C@H](CO)N[C@H]3C#N)C=C2)=C(F)C=1
Formula:	C₁₇H₁₅FN₂O
M.Wt:	282.312207460403
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

A small-molecule, allosteric inhibitor of Mycobacterium tuberculosis tryptophan synthase (TrpAB); binds at the TrpAB α-β-subunit interface with IC50 of 70.9 nM and 22.6 nM for α-subunit and β-subunit, respectively; highly effective in vivo.

MSDS

COA

LOT NO.	DOWNLOAD

2018-0101

Cat. No.	Product name	Field of application
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DC75641	GENZ-644282 TFA salt	Genz-644282, also known as SAR402674, is a non-camptothecin inhibitor of topoisomerase I with potential antineoplastic activity. Topoisomerase I inhibitor Genz-644282 binds to and inhibits the enzyme topoisomerase I, which may result in the inhibition of repair of single-strand DNA breaks, DNA replication, and tumor cell growth in susceptible tumor cell populations.
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DC74748	O4I4	O4I4 (compound 23) is a OCT4-inducing compound with metabolical stability.
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