CDE 096| CAS 1228357-04-7

Cas No.:	1228357-04-7
Chemical Name:	3-(((3-(Trifluoromethyl)phenoxy)carbonyl)amino)propane-1,2-diyl bis(3,4,5-trihydroxybenzoate)
Synonyms:	3-(((3-(trifluoromethyl)phenoxy)carbonyl)amino)propane-1,2-diyl bis(3,4,5-trihydroxybenzoate);CDE-096;[3-[[3-(trifluoromethyl)phenoxy]carbonylamino]-2-(3,4,5-trihydroxybenzoyl)oxypropyl] 3,4,5-trihydroxybenzoate;GLXC-04309;1228357-04-7;CS-0078249;1-({[3-(trifluoromethyl)phenoxy]carbonyl}amino)-3-(3,4,5-trihydroxybenzoyloxy)propan-2-yl 3,4,5-trihydroxybenzoate;OXWKLJPAKUDPJY-UHFFFAOYSA-N;EX-A5191;AKOS040746678;HY-120516;SCHEMBL13286848;3-(((3-(Trifluoromethyl)phenoxy)carbonyl)amino)-propane-1,2-diyl bis(3,4,5-trihydroxybenzoate)
SMILES:	FC(C1C=CC=C(C=1)OC(NCC(COC(C1C=C(C(=C(C=1)O)O)O)=O)OC(C1C=C(C(=C(C=1)O)O)O)=O)=O)(F)F
Formula:	C₂₅H₂₀F₃NO₁₂
M.Wt:	583.421018600464
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

A selective, reversible, high-affinity PAI-1 inhibitor that prevents PAI-1 from inactivating tPA and uPA with similar potency (IC50=30 and 25 nM, respectively); shows ineffective against two closely related serpins, antithrombin and α1-PI; blocks PAI-1 binding to vitronectin with IC50 of 22 nM.

MSDS

COA

LOT NO.	DOWNLOAD

2018-0101

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