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Olinone

  Cat. No.:  DC23372   Featured
Chemical Structure
1770789-37-1
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More than 5000 active chemicals with high quality for research!
Field of application
Olinone is a selective inhibitor for the BET BRD1 with Kd of 3.4/3.7/8.6 uM for BRD4-BrD1/BRD3-BrD1/BRD2-BrD1, respectively, shows high selectivity over BET BRD2 (Kd>300 uM).
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 1770789-37-1
Chemical Name: N-[4-(1-Oxo-1,2,3,4-Tetrahydro-5h-Pyrido[4,3-B]indol-5-Yl)butyl]acetamide
Synonyms: Olinone;N-[4-(1-Oxo-1,2,3,4-Tetrahydro-5h-Pyrido[4,3-B]indol-5-Yl)butyl]acetamide;N-[4-(1-Oxo-1,2,3,4-tetrahydro-pyrido[4,3-b]indol-5-yl)-butyl]-acetamide;AOB6713;SYN5213;BDBM50148603;J3.654.693J;Q27453447;N-[4-(1-oxo-3,4-dihydro-2H-pyrido[4,3-b]indol-5-yl)butyl]acetamide;N-[4-(1-Oxo-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole-5-yl)butyl]acetamide;30M
SMILES: O=C1C2C3=C([H])C([H])=C([H])C([H])=C3N(C([H])([H])C([H])([H])C([H])([H])C([H])([H])N([H])C(C([H])([H])[H])=O)C=2C([H])([H])C([H])([H])N1[H]
Formula: C17H21N3O2
M.Wt: 299.3675
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: Olinone is a selective inhibitor for the BET BRD1 with Kd of 3.4/3.7/8.6 uM for BRD4-BrD1/BRD3-BrD1/BRD2-BrD1, respectively, shows high selectivity over BET BRD2 (Kd>300 uM).
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
2018-0101
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