Cas No.: | 2092923-21-0 |
Chemical Name: | 5H-Imidazo[2,1-a]isoindol-5-one, 9b-(4-chloro-3-methylphenyl)-1-(3,4-difluorobenzoyl)-1,2,3,9b-tetrahydro-, (9bS)- |
Synonyms: | VU6008667 |
Formula: | C24H17ClF2N2O2 |
M.Wt: | 438.859 |
Purity: | >98% |
Sotrage: | 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO |
Description: | VU 6008667 is a potent, highly selective M5 negative allosteric modulator with IC50 of 1.2 uM; shows high CNS penetration, excellent selectivity versus M1-4 and the desired short half-life (t1/2=2.3h) in rats. |