Cas No.: | 145231-45-4 |
Chemical Name: | Carbamimidothioic acid, [(4-chlorophenyl)methyl]-, 3-(1H-imidazol-4-yl)propyl ester (9CI) |
Synonyms: | VUF-9153;VUF9153 |
SMILES: | Br.Br.N/C(=N/CC1C=CC(Cl)=CC=1)/SCCCC1=CN=CN1 |
Formula: | C14H17ClN4S |
M.Wt: | 308.828 |
Purity: | >98% |
Sotrage: | 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO |
Description: | Clobenpropit (VUF-9153) is a highly potent histamine H3 antagonist/inverse agonist with pA2 value of 9.93, also displays partial agonist activity at H4 receptors; increases brain histidine decarboxylase activity dose dependently, inhibits electrically induced convulsions in mice. |