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VU0155094(ML-397)

  Cat. No.:  DC23497   Featured
Chemical Structure
731006-86-3
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More than 5000 active chemicals with high quality for research!
Field of application
VU0155094 is a potent, selective pan-Group III mGlu positive allosteric modulator with IC50 of 3.43/1.5/0.93 uM for mGlu8/7/4, respectively.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 731006-86-3
Chemical Name: Methyl 4-[3-[2-(4-acetamidophenyl)sulfanylacetyl]-2,5-dimethylpyrrol-1-yl]benzoate
Synonyms: ML397;ML 397;methyl 4-[3-[2-(4-acetamidophenyl)sulfanylacetyl]-2,5-dimethylpyrrol-1-yl]benzoate;MLS000418059;GTPL10238;HMS2553G20;BDBM50283491;SMR000264819;VU0155094;VU 0155094;VU0155094-4;VU0155094-5;Z25065658;methyl 4-(3-(2-((4-acetamidophenyl)thio)acetyl)-2,5-dimethyl-1h-pyrrol-1-yl) benzoate;methyl 4-(3-(2-((4-acetamidophenyl)thio)acetyl)-2,5-dimethyl-1H-pyrrol-1-yl)benzoate;methyl 4
SMILES: S(C1C([H])=C([H])C(=C([H])C=1[H])N([H])C(C([H])([H])[H])=O)C([H])([H])C(C1C([H])=C(C([H])([H])[H])N(C2C([H])=C([H])C(C(=O)OC([H])([H])[H])=C([H])C=2[H])C=1C([H])([H])[H])=O
Formula: C24H24N2O4S
M.Wt: 436.5234
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: VU0155094 is a potent, selective pan-Group III mGlu positive allosteric modulator with IC50 of 3.43/1.5/0.93 uM for mGlu8/7/4, respectively; displays >30-fold selectivity over groups I and II mGlus (mGlu1/2/3/5/6).
References: References 1. Jalan-Sakrikar N, et al. ACS Chem Neurosci. 2014 Dec 17;5(12):1221-37. View Related Products by Target mGluR
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
2018-0101
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