Cas No.: | 935868-50-1 |
Chemical Name: | (R)-1-(2-(3,5-dichlorophenyl)pyridin-3-yl)-2,2-di(pyridin-3-yl)ethan-1-ol |
Synonyms: | MK1832 |
Formula: | C23H17Cl2N3O |
M.Wt: | 422.309 |
Purity: | >98% |
Sotrage: | 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO |
Description: | MK-1832 is a potent, selective Kv1.5 inhibitor with IC50 of 86 nM, exhibits improved selectivity for IKur over IKs (>3000-fold) compares with MK-0448 (70-fold), also exhibits an improved preclinical pharmacokinetic profile. |