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LY2452473

  Cat. No.:  DC23720   Featured
Chemical Structure
1029692-15-6
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More than 5000 active chemicals with high quality for research!
Field of application
LY2452473 is an orally bioavailable, selective androgen receptor modulator (SARM).
Cas No.: 1029692-15-6
Chemical Name: LY2452473
Synonyms: LY-2452473;Isopropyl (2S)-7-Cyano-4-(pyridin-2-ylmethyl)-1,2,3,4-tetrah;Isopropyl (2S)-7-Cyano-4-(pyridin-2-ylmethyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-2-ylcarbama;Isopropyl (2S)-7-Cyano-4-(pyridin-2-ylmethyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-2-ylcarbamate;(S)-ISOPROPYL (7-CYANO-4-(PYRIDIN-2-YLMETHYL)-1,2,3,4-TETRAHYDROCYCLOPENTA[B]INDOL-2-YL)CARBAMATE;LY2452473;XKW9MYF94Y;isopropyl (S)-(7-cyano-4-(pyridin-2-ylmethyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-2-yl)carbamate;DB12573;Carbamic acid, N-((2S)-7-cyano-1,2,3,4-tetrahydro-4
SMILES: O(C(C)C)C(N[C@H]1CC2C3C=C(C#N)C=CC=3N(CC3C=CC=CN=3)C=2C1)=O
Formula: C22H22N4O2
M.Wt: 374.435684680939
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: LY2452473 (TT 701;OPK 88004) is an orally bioavailable selective androgen receptor modulator (SARM) being developed for the treatment of disorders related to hypogonadism; has the potential advantage of eliciting androgen receptor specificity and tissue selectivity to produce the beneficial effects of testosterone on bone, muscle, and improvements in erectile function over a PDE5i alone, with minimal steroid-related adverse effects.Prostate CancerPhase 2 Clinical
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
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