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MAP4K4-IN-17

  Cat. No.:  DC23814   Featured
Chemical Structure
1811510-58-3
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More than 5000 active chemicals with high quality for research!
Field of application
MAP4K4-IN-17 is a potent and highly selective MAP4K4 inhibitor with IC50 of 14.9 nM, showes improved overall drug-like properties compared to PF-06260933.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 1811510-58-3
Chemical Name: MAP4K4-IN-17
Synonyms: 5-(6-amino-5-(4-chlorophenyl)pyridin-3-yl)pyrimidin-2-amine
SMILES: NC1=NC=C(C2=CC(C3=CC=C(Cl)C=C3)=C(N)N=C2)C=N1
Formula: C15H12ClN5
M.Wt: 297.746
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: MAP4K4-IN-17 is a potent and highly selective MAP4K4 inhibitor with IC50 of 14.9 nM, showes improved overall drug-like properties compared to PF-06260933; a lead compound for advanced preclinical development.
References: References 1. Ammirati M, et al. ACS Med Chem Lett. 2015 Oct 6;6(11):1128-33. View Related Products by Target MAP4K
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
2018-0101
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