Cas No.: | 912656-34-9 |
Chemical Name: | Spiro[furo[2,3-f]-1,3-benzodioxole-7(6H),3'-[3H]indol]-2'(1'H)-one, 1'-pentyl- |
Synonyms: | XEN907;XEN 907 |
SMILES: | O=C1N(C2C=CC=CC=2C21C1C=C3C(=CC=1OC2)OCO3)CCCCC |
Formula: | C21H21NO4 |
M.Wt: | 351.3958 |
Purity: | >98% |
Sotrage: | 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO |
Description: | A potent, selective NaV1.7 blocker with IC50 of 3 nM; shows no significant activity at 10 uM against a broad panel of 63 receptors and transporters; has no cytotoxic and favourable hepatocyte metabolic stability for both human and dog,PainPreclinical |