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GNE-616

  Cat. No.:  DC26078   Featured
Chemical Structure
2244895-99-4
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More than 5000 active chemicals with high quality for research!
Field of application
GNE-616 (GNE616) is a highly potent, metabolically stable, subtype selective inhibitor of Nav1.7 with Ki of 0.79 nM (hNav1.7).
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 2244895-99-4
Chemical Name: 2H-1-Benzopyran-7-sulfonamide, 6-fluoro-3,4-dihydro-4-[(2S,4R)-2-(2-pyridinyl)-4-(trifluoromethyl)-1-piperidinyl]-N-4-pyrimidinyl-, (4S)-
Synonyms: 2H-1-Benzopyran-7-sulfonamide, 6-fluoro-3,4-dihydro-4-[(2S,4R)-2-(2-pyridinyl)-4-(trifluoromethyl)-1-piperidinyl]-N-4-pyrimidinyl-, (4S)-
SMILES: C1OC2=CC(S(NC3C=CN=CN=3)(=O)=O)=C(F)C=C2[C@@H](N2CC[C@@H](C(F)(F)F)C[C@H]2C2=NC=CC=C2)C1
Formula: C24H23F4N5O3S
M.Wt: 537.53
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
Cat. No. Product name Field of application
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