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PF-05198007

  Cat. No.:  DC26091   Featured
Chemical Structure
1235406-19-5
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More than 5000 active chemicals with high quality for research!
Field of application
PF-05198007 is a potent, state-dependent, subtype selective Nav1.7 inhibitor with IC50 of 9 nM, no significant activity against Nav1.5 (IC50>10 uM).
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 1235406-19-5
Chemical Name: 4-(2-(3-Amino-1H-pyrazol-4-yl)-4-(trifluoromethyl)phenoxy)-5-chloro-2-fluoro-N-(thiazol-4-yl)benzenesulfonamide
Synonyms: 4-(2-(3-Amino-1H-pyrazol-4-yl)-4-(trifluoromethyl)phenoxy)-5-chloro-2-fluoro-N-(thiazol-4-yl)benzenesulfonamide;BDBM50257214;4-[2-(3-amino-1h-pyrazol-4-yl)-4-(trifluoromethyl)phenoxy]-5-chloro-2-fluoro-n-1,3-thiazol-4-ylbenzenesulfonamide;4-[2-(5-amino-1H-pyrazol-4-yl)-4-(trifluoromethyl)phenoxy]-5-chloro-2-fluoro-N-(1,3-thiazol-4-yl)benzenesulfonamide;PF-05198007
SMILES: ClC1C=C(C(=CC=1OC1=CC=C(C(F)(F)F)C=C1C1C=NNC=1N)F)S(NC1=CSC=N1)(=O)=O
Formula: C19H12ClF4N5O3S2
M.Wt: 533.906893730164
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
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