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Poloppin

  Cat. No.:  DC26116   Featured
Chemical Structure
683808-78-8
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More than 5000 active chemicals with high quality for research!
Field of application
Poloppin is a cell-active, small molecule inhibitor of protein-protein interaction via the Polo-box domain (PBD) of the mitotic Polo-like kinase (PLK) with IC50 of 26.9 uM (PLK1) in FP assays.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 683808-78-8
Chemical Name: Poloppin
Synonyms: Poloppin;3-(5-(4-Bromophenyl)-1-(2-(trifluoromethyl)phenyl)-1H-pyrrol-2-yl)propanoic acid;3-{5-(4-bromophenyl)-1-[2-(trifluoromethyl)phenyl]-1H-pyrrol-2-yl}propanoic acid;STK278324;5-(4-Bromophenyl)-1-[2-(trifluoromethyl)phenyl]-1H-pyrrole-2-propanoic acid;Polo protein-protein interaction inhibitor
SMILES: BrC1C=CC(=CC=1)C1=CC=C(CCC(=O)O)N1C1C=CC=CC=1C(F)(F)F
Formula: C20H15BrF3NO2
M.Wt: 438.237815141678
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
Cat. No. Product name Field of application
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