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GPR52-IN-43(CAY10786)

  Cat. No.:  DC60162   Featured
Chemical Structure
1239987-91-7
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More than 5000 active chemicals with high quality for research!
Field of application
GPR52-IN-43(CAY10786) is a novel GPR52 antagonist, reducing mHTT levels by targeting GPR52 and promoting survival of mouse primary striatal neurons, and also reducing HD-related phenotypes in HdhQ140.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 1239987-91-7
Chemical Name: (2E)-5-Phenyl-1-(2-thienyl)-2-penten-1-one
Synonyms: (2E)-5-phenyl-1-(2-thienyl)-2-penten-1-one;(E)-5-phenyl-1-thiophen-2-ylpent-2-en-1-one
SMILES: S1C([H])=C([H])C([H])=C1C(/C(/[H])=C(\[H])/C([H])([H])C([H])([H])C1C([H])=C([H])C([H])=C([H])C=1[H])=O
Formula: C15H14Os
M.Wt: 242.3361
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: GPR52-IN-43(CAY10786) is a novel GPR52 antagonist, reducing mHTT levels by targeting GPR52 and promoting survival of mouse primary striatal neurons, and also reducing HD-related phenotypes in HdhQ140.
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