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Eprobemide (LIS 630)

  Cat. No.:  DC12311   Featured
Chemical Structure
87940-60-1
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More than 5000 active chemicals with high quality for research!
Field of application
Eprobemide is a non-competitive reversible inhibitor of monoamine oxidase A.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 87940-60-1
Chemical Name: LIS 630；LIS-630；LIS630
SMILES: O=C(NCCCN1CCOCC1)C2=CC=C(Cl)C=C2
Formula: C14H19ClN2O2
M.Wt: 282.77
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: Eprobemide is a non-competitive reversible inhibitor of monoamine oxidase A.
Target: Monoamine oxidase A[1][2]
In Vitro: Eprobemide is a pharmaceutical drug that is used as an antidepressant. Eprobemide is a non-competitive reversible inhibitor of monoamine oxidase A that exhibits selective action on serotonin deamination[1][2].
References: [1]. Gol'dina OA, et al. The action of befol and its derivatives on monoamine oxidase of different origins. Biull Eksp Biol Med. 1991 Mar;111(3):279-80. [2]. Donskaya, et al. Antidepressant Befol Synthesized Via Interaction of 4-Chloro-N-(3-chloropropyl)benzamide with Morpholine. Pharmaceutical Chemistry Journal, 2004 Jun; 38(7): 381-384.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
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