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GOT1 inhibitor 2c

  Cat. No.:  DC12542   Featured
Chemical Structure
732973-87-4
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More than 5000 active chemicals with high quality for research!
Field of application
GOT1 inhibitor 2c is a first-in-class, non-covalent inhibitor of glutamate oxaloacetate transaminase 1 (GOT1) with IC50 of 8.2 uM..
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 732973-87-4
Chemical Name: N-(4-chlorophenyl)-4-(1H-indol-4-yl)piperazine-1-carboxamide
SMILES: O=C(N1CCN(C2=CC=CC3=C2C=CN3)CC1)NC4=CC=C(Cl)C=C4
Formula: C19H19ClN4O
M.Wt: 354.83
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Publication: 1. Anglin J, et al. Bioorg Med Chem Lett. 2018 Sep 1;28(16):2675-2678.
Description: GOT1 inhibitor 2c is a first-in-class, non-covalent inhibitor of glutamate oxaloacetate transaminase 1 (GOT1) with IC50 of 8.2 uM.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
2018-0101
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