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GSK-2894631A(HPGDS inhibitor 2)

  Cat. No.:  DC22317   Featured
Chemical Structure
2101626-26-8
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More than 5000 active chemicals with high quality for research!
Field of application
GSK-2894631A,GSK 2894631A，GSK2894631A
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 2101626-26-8
SMILES: C1C2=CC=C(OC(F)F)C=C2N=CC=1C(N[C@@H]1CC[C@@H](C(O)(C)C)CC1)=O
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: GSK-2894631A(HPGDS inhibitor 2) is a highly potent and selective hematopoietic prostaglandin D synthase (H-PGDS) inhibitor with an IC50 of 9.9 nM[1].
Target: IC50: 9.9 nM (H-PGDS)[1]
References: [1]. Deaton DN, et al. The discovery of quinoline-3-carboxamides as hematopoietic prostaglandin D synthase (H-PGDS) inhibitors. Bioorg Med Chem. 2019 Apr 15;27(8):1456-1478.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
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