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Protein kinase inhibitor 1

  Cat. No.:  DC10898   Featured
Chemical Structure
1365986-44-2
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More than 5000 active chemicals with high quality for research!
Field of application
It is a novel inhibitor of HIPK2 with an IC50 of 74 nM and Kd of 9.5 nM.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 1365986-44-2
Chemical Name: Protein kinase inhibitor 1
Synonyms: Protein kinase inhibitors 1;Protein kinase inhibitors 1 hydrochlorid (1365986-44-2(free base));Protein kinase inhibitor 1
SMILES: Cl.S1C(NC(/C/1=C/C1=CNC(C(=C1)C1=CN=C(C=C1)N1CCNCC1)=O)=O)=O
Formula: C18H18ClN5O3S
M.Wt: 383.430
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: Protein kinase inhibitors 1 is a novel inhibitor of HIPK2 with an IC50 of 74 nM and Kd of 9.5 nM.
References: [1]. Miduturu CV, et al. High-throughput kinase profiling: a more efficient approach toward the discovery of new kinaseinhibitors. Chem Biol. 2011 Jul 29;18(7):868-79.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
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