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Indibulin

  Cat. No.:  DC31248   Featured
Chemical Structure
204205-90-3
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More than 5000 active chemicals with high quality for research!
Field of application
Indibulin is a synthetic small molecule with antimitotic and potential antineoplastic activities. Indibulin binds to a site on tubulin that is different from taxane- or Vinca alkaloid-binding sites, destabilizing tubulin polymerization and inducing tumor cell cycle arrest and apoptosis. This agent has been shown to be active against multidrug-resistant (MDR) and taxane- resistant tumor cell lines. Check for active clinical trials or closed clinical trials using this agent. (NCI Thesaurus).
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 204205-90-3
Chemical Name: 2-(1-(4-chlorobenzyl)-1H-indol-3-yl)-2-oxo-N-(pyridin-4-yl)acetamide
Synonyms: ZIO-301；ZERO/005632；ZINC01996564；d-24851; D-24851；NCGC00160428-01.
SMILES: O=C(NC1=CC=NC=C1)C(C2=CN(CC3=CC=C(Cl)C=C3)C4=C2C=CC=C4)=O
Formula: C22H16ClN3O2
M.Wt: 389.83
Purity: 98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
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