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KDM5A covalent inhibitor N73

  Cat. No.:  DC12520  
Chemical Structure
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More than 5000 active chemicals with high quality for research!
Field of application
KDM5A covalent inhibitor N73 is the the isopropyl ester derivative of N71, an irreversible KDM5A inhibitor (IC50=0.22 uM) that covalently interacts with Cys481, >20-fold selectivity over KDM4A..
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.:
Chemical Name: isopropyl (E)-2-((3-(4-(dimethylamino)but-2-enamido)phenyl)(2-(piperidin-1-yl)ethoxy)methyl)thieno[3,2-b]pyridine-7-carboxylate
SMILES: C12C=C(C(C3=CC=CC(NC(=O)/C=C/CN(C)C)=C3)OCCN3CCCCC3)SC1=C(C(OC(C)C)=O)C=CN=2
Formula: C31H40N4O4S
M.Wt: 564.745
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
Cat. No. Product name Field of application
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Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.
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