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NAV26

  Cat. No.:  DC34303   Featured
Chemical Structure
1198160-14-3
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More than 5000 active chemicals with high quality for research!
Field of application
NAV 26 (compound 26) is a selective voltage-gated sodium channel Nav1.7 blocker with an IC50 of 0.37 μM. NAV 26 can be used for pain research.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 1198160-14-3
Chemical Name: 2,3-Dihydro-3-oxo-2-(tetrahydro-2H-pyran-4-yl)-N-4-(trifluoromethoxy)phenylmethyl-1H-Isoindole-1-carboxamide
Synonyms: 2,3-Dihydro-3-oxo-2-(tetrahydro-2H-pyran-4-yl)-N-[[4-(trifluoromethoxy)phenyl]methyl]-1H-Isoindole-1-carboxamide;NAV 26;BDBM50395368;2-(Oxan-4-yl)-3-oxo-N-[[4-(trifluoromethoxy)phenyl]methyl]-1H-isoindole-1-carboxamide
SMILES: FC(OC1C=CC(=CC=1)CNC(C1C2C=CC=CC=2C(N1C1CCOCC1)=O)=O)(F)F
Formula: C22H21F3N2O4
M.Wt: 434.408356428146
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
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COA
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Cat. No. Product name Field of application
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DC75641 GENZ-644282 TFA salt Genz-644282, also known as SAR402674, is a non-camptothecin inhibitor of topoisomerase I with potential antineoplastic activity. Topoisomerase I inhibitor Genz-644282 binds to and inhibits the enzyme topoisomerase I, which may result in the inhibition of repair of single-strand DNA breaks, DNA replication, and tumor cell growth in susceptible tumor cell populations.
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DC74646 EB-PSMA-617 EB-PSMA-617 is an Evans blue-modified prostate-specific membrane antigen (PSMA) 617 ligand for making 177Lu-EB-PSMA, which is potential useful for Metastatic Castration-Resistant Prostate Cancer.
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