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Omadacycline (tosylate)

  Cat. No.:  DC10365   Featured
Chemical Structure
1075240-43-5
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More than 5000 active chemicals with high quality for research!
Field of application
Omadacycline is novel, aminomethyl tetracycline antibiotic being developed for the treatment of community-acquired bacterial infections.
Cas No.: 1075240-43-5
Chemical Name: Omadacycline (tosylate)
Synonyms: Omadacycline (tosylate);Amadacycline tosylate;PTK 0796 tosylate;PTK-0796 tosylate
SMILES: CC1C=CC(S(=O)(O)=O)=CC=1.O=C(N)C1C(=O)C2(O)C(O)=C3C(=O)C4C(CC3([H])CC2([H])C(N(C)C)C=1O)=C(N(C)C)C=C(CNCC(C)(C)C)C=4O
Formula: C36H48N4O10S
M.Wt: 728.852128982544
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Publication: [1]. Schmitz J, Holzgrabe U. Amadacyclin - a new tetracycline antibiotic in the pipeline. Pharm Unserer Zeit. 2010 Mar;39(2):94-5.
Description: Omadacycline tosylate is a new tetracycline antibiotic in the pipeline, which can inhibit the 30s subunit of bacterial ribosome.
Target: Antibacterial
In Vivo: Clinical trial: Phase III Study to Compare the Safety and Efficacy of PTK-0796 in Patients With Complicated Skin and Skin Structure Infection (CSSSI).
References: [1]. Schmitz J, Holzgrabe U. Amadacyclin - a new tetracycline antibiotic in the pipeline. Pharm Unserer Zeit. 2010 Mar;39(2):94-5.
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