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PD-166793

  Cat. No.:  DC37910   Featured
Chemical Structure
199850-67-4
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More than 5000 active chemicals with high quality for research!
Field of application
PD-166793 is a cell-permeable biphenylsulfonylvaline compound that acts as a potent inhibitor against MMP-2, -3, and -13 (IC50 = 47, 12, and 8 nM, respectively) and a weaker inhibitor against AMP deaminase (20% inhibition at 0.1 μM), MMP-1, -7, -9, and -14 (IC50 = 6.1, 7.2, 7.9, and 0.24 μM, respectively). Shown to offer therapeutic benefits in vivo in various animal models of heart failure and diabetes.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 199850-67-4
Chemical Name: ((4'-bromo-[1,1'-biphenyl]-4-yl)sulfonyl)-L-valine
Synonyms: PD-166793; PD 166793; PD166793; PD-166793-0000;
SMILES: CC(C)[C@@H](C(O)=O)NS(=O)(C1=CC=C(C2=CC=C(Br)C=C2)C=C1)=O
Formula: C17H18BrNO4S
M.Wt: 412.29
Purity: 98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
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COA
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