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PKC-theta inhibitor

  Cat. No.:  DC26157   Featured
Chemical Structure
736048-65-0
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More than 5000 active chemicals with high quality for research!
Field of application
PKC-theta inhibitor is a selective PKC-θinhibitor, with an IC50 of 12 nM.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 736048-65-0
SMILES: FC(F)(F)OC1=CC=CC=C1CNC2=NC=C([N+]([O-])=O)C(NCC3CCC(CN)CC3)=N2
Formula: C20H25F3N6O3
M.Wt: 454.45
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
Description: PKC-theta inhibitor is a selective PKC-θinhibitor, with an IC50 of 12 nM.
Target: PKCθ:12 nM (IC50)
References: [1]. Cywin CL, et al. Discovery of potent and selective PKC-theta inhibitors. Bioorg Med Chem Lett. 2007 Jan 1;17(1):225-30.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
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