PKCiota-IN-49|cas 2230055-52-2|DC Chemiclas

Cas No.:	2230055-52-2
Chemical Name:	PKCiota-IN-49
Synonyms:	PKCiota-IN-49;PKCiota-IN-2
SMILES:	C1C2=C(C=C(OC)C(C3=C4N(N=C3)C=CC(C3C=CN=C5NC=CC5=3)=C4)=C2)CCN1
Formula:	C₂₄H₂₁N₅O
M.Wt:	395.46
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

PKCiota-IN-2 is a potent PKCiota (PKC-ι) inhibitor with an IC50 of 2.8 nM. PKCiota-IN-2 also inhibits PKC-α and PKC-ε with IC50s of 71 nM and 350 nM, respectively.

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