PL-017|CAS 83397-56-2|DC Chemicals

Cas No.:	83397-56-2
Chemical Name:	PL-017
Synonyms:	YP-{N(Me)Phe}-P-NH2
Formula:	C₂₉H₃₇N₅O₅
M.Wt:	535.63
Sotrage:	Please store the product under the recommended conditions in the Certificate of Analysis.

Cat. No.	Product name	Field of application
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DC45826	BMS-986121	BMS-986121 is a positive allosteric modulator (PAM) of the μ opioid receptor extracted from patent WO2014107344. BMS-986121 is built on a chemical scaffold representing a new chemotype for μ receptor PAMs.
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DC45524	Deltorphin 2 TFA	Deltorphin 2 TFA is a selective peptide agonist for the δ opioid receptor.
DC44749	6'-GNTI dihydrochloride	6'-GNTI dihydrochloride, a κ-opioid receptor (KOR) agonist, displays bias toward the activation of G protein-mediated signaling over β-arrestin2 recruitment. 6'-GNTI 6'-GNTI dihydrochloride only activates the Akt pathway in striatal neurons.
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DC42315	Cebranopadol ((1α,4α)stereoisomer)	Cebranopadol ((1α,4α)stereoisomer) is a stereoisomer of cebranopadol. Cebranopadol is a potent agonist activity on ORL-1.
DC41867	Dynorphin A (1-8)	Dynorphin A (1-8) is the predominant opioid peptide identified in placental tissue extracts. Dynorphin A (1-8) is the most likely natural ligand of the kappa receptor. The binding of 3H-Bremazocine to the purified kappa receptor is inhibited by Dynorphin A (1-8) (IC50=303 nM).