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Pimavanserin tartrate

  Cat. No.:  DC32110   Featured
Chemical Structure
706782-28-7
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Field of application
Pimavanserin, also known as ACP-103, is a non-dopaminergic atypical antipsychotic for the treatment of Parkinson's disease psychosis and schizophrenia. Pimavanserin has a unique mechanism of action relative to other antipsychotics, behaving as a selective inverse agonist of the serotonin 5-HT2A receptor, with 40-fold selectivity for this site over the 5-HT2C receptor and no significant affinity or activity at the 5-HT2B receptor or dopamine receptors. It was approved by the FDA to treat hallucinations and delusions associated with psychosis experienced by some people with Parkinson's disease on April 29, 2016.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 706782-28-7
Chemical Name: Pimavanserin Tartrate
Synonyms: Pimavanserin Tartrate;Unii-na83F1sjsr
SMILES: O=C(NCC1=CC=C(OCC(C)C)C=C1)N(CC2=CC=C(F)C=C2)C3CCN(C)CC3.O=C(O)[C@H](O)[C@@H](O)C(O)=O.O=C(NCC4=CC=C(OCC(C)C)C=C4)N(CC5=CC=C(F)C=C5)C6CCN(C)CC6
Formula: C54H74F2N6O10
M.Wt: 1005.19638204575
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
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MSDS_14422_DC32110_706782-28-7
COA
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