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SSR180711 hydrochloride

  Cat. No.:  DC41121  
Chemical Structure
446031-79-4
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More than 5000 active chemicals with high quality for research!
Field of application
SSR180711 hydrochloride is an orally active, selective and reversible α7 acetylcholine nicotinic receptor (n-AChRs) partial agonist. SSR180711 hydrochloride can act on rat α7 n-AChR (Ki=22 nM; IC50=30 nM) and human α7 n-AChR (Ki=14 nM; IC50=18 nM). SSR180711 hydrochloride increases glutamatergic neurotransmission, ACh release and long-term potentiation (LTP) in the hippocampus.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 446031-79-4
Chemical Name: SSR180711 hydrochloride
SMILES: O=C(N1CCN2CCC1CC2)OC3=CC=C(Br)C=C3.[H]Cl
Formula: C14H18BrClN2O2
M.Wt: 361.66
Sotrage: Please store the product under the recommended conditions in the Certificate of Analysis.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
Cat. No. Product name Field of application
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DC46640 Sulfoxaflor Sulfoxaflor is a sulfoximine insecticide and is an agonist of nAChR1 and nAChR2 subtypes. Sulfoxaflor is used for the control of sap-feeding insects such as Myzus persicae, Aphis gossypii, Bemissia tabaci and Nilaparvata lugens.
DC46496 TQS TQS is a α7 nicotinic acetylcholine receptor (nAChR) positive allosteric modulator. TQS can be used for the research of neuroinflammatory pain.
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