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Tracazolate hydrochloride

  Cat. No.:  DC41239  
Chemical Structure
1135210-68-2
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More than 5000 active chemicals with high quality for research!
Field of application
Tracazolate (ICI 136753) hydrochloride is a potent GABAA receptor modulator. Tracazolate hydrochloride has selectivity for β3 and potentiates α1β1γ2s (EC50=13.2 μM), α1β3γ2 (EC50=1.5 μM). Tracazolate hydrochloride has the potency (EC50) determined by the nature of the third subunit (γ1-3, δ, ε) within the receptor complex. Tracazolate hydrochloride possesses anxiolytic and anticonvulsant activity.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 1135210-68-2
Chemical Name: Tracazolate HCl
SMILES: O=C(C1=C(C)N=C(N(CC)N=C2)C2=C1NCCCC)OCC.[H]Cl
Formula: C16H25ClN4O2
M.Wt: 340.85
Sotrage: Please store the product under the recommended conditions in the Certificate of Analysis.
MSDS
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MSDS_24252_DC41239_1135210-68-2
COA
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Cat. No. Product name Field of application
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