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URB-937

  Cat. No.:  DC39032   Featured
Chemical Structure
1357160-72-5
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More than 5000 active chemicals with high quality for research!
Field of application
URB937 is a potent fatty acid amide hydrolase (FAAH) inhibitor (IC50 = 26.8 nM, in vitro) that does not penetrate the blood-brain barrier, thus preventing arachidonoyl ethanolamidedeactivation only in peripheral tissues.
Chemicals PropertiesBiological activity Related products COA MSDS Datasheet
Cas No.: 1357160-72-5
Chemical Name: Cyclohexylcarbamic acid 3′–carbamoyl–6–hydroxybiphenyl–3–yl ester;3'-Carbamoyl-6-hydroxybiphenyl-3-yl cyclohexylcarbamate
Synonyms: URB 937;URB937;URB-937
SMILES: NC(C1=CC=CC(C2C=C(OC(NC3CCCCC3)=O)C=CC=2O)=C1)=O
Formula: C20H22N2O4
M.Wt: 354.399685382843
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Publication: [1]. Jason R Clapper, et al. Anandamide suppresses pain initiation through a peripheral endocannabinoid mechanism. Nat Neurosci. 2010 Oct;13(10):1265-70.
Description: URB937 is a potent fatty acid amide hydrolase (FAAH) inhibitor (IC50 = 26.8 nM, in vitro) that does not penetrate the blood-brain barrier, thus preventing arachidonoyl ethanolamidedeactivation only in peripheral tissues.
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