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AZ3976

  Cat. No.:  DC42708   Featured
Chemical Structure
1418747-15-5
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More than 5000 active chemicals with high quality for research!
Field of application
AZ3976 is a selective PAI-1 inhibitor that exhibits potent profibrinolytic effects, with IC50 values of 26 μM (chromogenic assay) and 16 μM (plasma clot lysis assay). Unlike conventional inhibitors, it does not target active PAI-1 but instead binds reversibly to the latent form, accelerating the transition of active PAI-1 to its inactive state.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 1418747-15-5
Chemical Name: 1-Boc-3-(4-Oxo-3,4-dihydro-pyrido[2,3-d]pyrimidin-2-ylamino)-azetidine
Synonyms: AZ3976;AZ-3976;AZ 3976
SMILES: O=C1C2=CC=CN=C2N=C(NC3CN(C(OC(C)(C)C)=O)C3)N1
Formula: C15H19N5O3
M.Wt: 317.34
Purity: >98%
Sotrage: 0°C (short term), -20°C (long term), desiccated
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
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