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Bexin-1

  Cat. No.:  DC42587   Featured
Chemical Structure
1172933-44-6
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More than 5000 active chemicals with high quality for research!
Field of application
Bexin-1 is a specific inhibitor that targets Munc13-4, a protein critical for regulated exocytosis, particularly in secretory cells such as immune cells (e.g., cytotoxic T lymphocytes, mast cells) and neuroendocrine cells. Munc13-4 plays a key role in vesicle priming and fusion with the plasma membrane, a process essential for the release of secretory granules containing hormones, neurotransmitters, or immune mediators.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 1172933-44-6
Chemical Name: Bexin-1
Synonyms: Bexin-1;N-(7-Chloro-4-methylbenzo[d]thiazol-2-yl)-N-(3-(dimethylamino)propyl)-1-ethyl-5-methyl-1H-pyrazole-3-carboxamide
SMILES: ClC1=CC=C(C)C2=C1SC(=N2)N(C(C1C=C(C)N(CC)N=1)=O)CCCN(C)C
Formula: C20H26ClN5Os
M.Wt: 419.971341609955
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
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