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Desketoraloxifene

  Cat. No.:  DC43269   Featured
Chemical Structure
216570-81-9
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More than 5000 active chemicals with high quality for research!
Field of application
Selective estrogen receptor modulator (SERM), inhibiting mammalian PLD (PLD1 and PLD2)
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 216570-81-9
Chemical Name: Desketoraloxifene
Synonyms: Desketoraloxifene;2-(4-hydroxyphenyl)-3-[4-(2-piperidin-1-ylethoxy)phenyl]-1-benzothiophen-6-ol;Desketoraloxifene (10);BDBM154519
SMILES: S1C2C=C(C=CC=2C(=C1C1C=CC(=CC=1)O)C1C=CC(=CC=1)OCCN1CCCCC1)O
Formula: C27H27NO3S
M.Wt: 445.573186159134
Purity: >98%
Sotrage: 0°C (short term), -20°C (long term), desiccated
MSDS
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MSDS_26894_DC43269_216570-81-9
COA
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Cat. No. Product name Field of application
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DC75868 AZ14133346 AZ14133346 (compound 36) is a potent and selective inhibitor of EGFR Exon20 insertions, with the IC50 of 85 nM. AZ14133346 plays an important role in cancer research.
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DC75816 Nisoxetine Nisoxetine acts as a highly selective and potent noradrenaline transporter (NET) antagonist, exhibiting a binding affinity (Kd) of 0.76 nM. In addition to its antidepressant properties, nisoxetine functions as a local anesthetic by inhibiting voltage-gated sodium channels. This dual pharmacological activity makes it a compound of interest for both neurological and pain management research.
DC75641 GENZ-644282 TFA salt Genz-644282, also known as SAR402674, is a non-camptothecin inhibitor of topoisomerase I with potential antineoplastic activity. Topoisomerase I inhibitor Genz-644282 binds to and inhibits the enzyme topoisomerase I, which may result in the inhibition of repair of single-strand DNA breaks, DNA replication, and tumor cell growth in susceptible tumor cell populations.
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DC74646 EB-PSMA-617 EB-PSMA-617 is an Evans blue-modified prostate-specific membrane antigen (PSMA) 617 ligand for making 177Lu-EB-PSMA, which is potential useful for Metastatic Castration-Resistant Prostate Cancer.
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