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G150

  Cat. No.:  DC42718   Featured
Chemical Structure
2369751-30-2
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More than 5000 active chemicals with high quality for research!
Field of application
G150 is a highly selective human cyclic GMP-AMP synthase (h-cGAS) inhibitor with an IC50 of 10.2 nM. G150 represses dsDNA-triggered interferon expression, and G150 can be used for the research of inflammatory.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 2369751-30-2
Chemical Name: G150
Synonyms: G150;1-[9-(6-aminopyridin-3-yl)-6,7-dichloro-1,3,4,5-tetrahydro-2H-pyrido[4,3-b]indol-2-yl]-2-hydroxyethan-1-one;s8944;JUJ;1-[9-(6-Aminopyridin-3-yl)-6,7-dichloro-1,3,4,5-tetrahydropyrido[4,3-b]indol-2-yl]-2-hydroxyethanone
SMILES: ClC1=C(C([H])=C(C2=C([H])N=C(C([H])=C2[H])N([H])[H])C2=C1N([H])C1C([H])([H])C([H])([H])N(C(C([H])([H])O[H])=O)C([H])([H])C=12)Cl
Formula: C18H16Cl2N4O2
M.Wt: 391.2512
Purity: >98%
Sotrage: 0°C (short term), -20°C (long term), desiccated
MSDS
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COA
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Cat. No. Product name Field of application
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