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GABAA receptor agent 2 TFA

  Cat. No.:  DC44910  
Chemical Structure
1781880-44-1
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More than 5000 active chemicals with high quality for research!
Field of application
GABAA receptor agent 2 TFA is a potent and high-affinity GABAA receptor antagonist with an IC50 of 24 nM (human α1β2γ2 GABAA-expressing tsA201 cells) and a Ki of 28 nM (rat GABAA receptors). GABAA receptor agent 2 TFA is inactive against four human GABA transporters (hGAT-1, hBGT-1, hGAT-2, and hGAT-3).
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 1781880-44-1
Chemical Name: GABAA receptor agent 2 TFA
SMILES: ON1N=CC(C2CCNCC2)=C1C3=CC(C4=CC=CC=C4)=CC=C3.OC(C(F)(F)F)=O
Formula: C22H22F3N3O3
M.Wt: 433.42
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
Cat. No. Product name Field of application
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