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GSK3987

  Cat. No.:  DC42709   Featured
Chemical Structure
264206-85-1
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More than 5000 active chemicals with high quality for research!
Field of application
GSK3987 functions as a dual agonist for both LXRα and LXRβ nuclear receptors, demonstrating potent activation with EC50 values of 50 nM (LXRα-SRC1) and 40 nM (LXRβ-SRC1). This compound effectively upregulates key metabolic regulators ABCA1 and SREBP-1c, while simultaneously promoting cholesterol efflux from cells and stimulating intracellular triglyceride deposition.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 264206-85-1
Chemical Name: 1-Benzyl-3-(4-methoxyanilino)-4-phenylpyrrole-2,5-dione
Synonyms: GSK3987
SMILES: O=C(C(NC1=CC=C(OC)C=C1)=C2C3=CC=CC=C3)N(CC4=CC=CC=C4)C2=O
Formula: C24H20N2O3
M.Wt: 384.44
Purity: >98%
Sotrage: 0°C (short term), -20°C (long term), desiccated
MSDS
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MSDS_26338_DC42709_264206-85-1
COA
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Cat. No. Product name Field of application
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