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KB-0742 dihydrochloride

  Cat. No.:  DC42486  
Chemical Structure
2416874-75-2
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Field of application
KB-0742 dihydrochloride is a potent, selective and orally active CDK9 inhibitor with an IC50 of 6 nM for CDK9/cyclin T1. KB-0742 dihydrochloride is selective for CDK9/cyclin T1 with >50-fold selectivity over other CDK kinases. KB-0742 dihydrochloride has potent anti-tumor activity.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 2416874-75-2
Chemical Name: KB-0742 HCl
Synonyms: KB-0742 dihydrochloride
SMILES: N[C@@H]1C[C@@H](NC2=CC(C(CC)CC)=NC3=CC=NN23)CC1.[H]Cl.[H]Cl
Formula: C16H27Cl2N5
M.Wt: 360.327
Sotrage: Please store the product under the recommended conditions in the Certificate of Analysis.
MSDS
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MSDS_26114_DC42486_2416874-75-2
COA
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Cat. No. Product name Field of application
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DC47130 CDK5-IN-1 CDK5-IN-1, a potent CDK5 inhibitor, is against CDK5 activity less than 10 nM. CDK5-IN-1 is used for kidney diseases research.
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