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MRTX 0902

  Cat. No.:  DC70046   Featured
Chemical Structure
2654743-22-1
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More than 5000 active chemicals with high quality for research!
Field of application
MRTX0902 is a potent SOS1 inhibitor with an IC50 of 46 nM (WO2021127429A1; Example 12-10).
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 2654743-22-1
Chemical Name: MRTX 0902
Synonyms: MRTX0902
SMILES: N#CC1=CC=CC([C@H](NC2=NN=C(C)C3=CN=C(N4CCOCC4)C=C32)C)=C1C
Formula: C22H24N6O
M.Wt: 388.475
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Publication: [1]. Matthew Arnold Marx, et al. Sos1 inhibitors. WO2021127429A1. [2]. Matthew Arnold Marx, et al. Sos1 inhibitors. WO2021127429A1.
Description: MRTX0902 is a potent SOS1 inhibitor with an IC50 of 46 nM (WO2021127429A1; Example 12-10).
References: [1]. Matthew Arnold Marx, et al. Sos1 inhibitors. WO2021127429A1. [2]. Matthew Arnold Marx, et al. Sos1 inhibitors. WO2021127429A1.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
Cat. No. Product name Field of application
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DC70046 MRTX 0902 MRTX0902 is a potent SOS1 inhibitor with an IC50 of 46 nM (WO2021127429A1; Example 12-10).
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