NCGC2955|CAS |DC Chemicals

Cas No.:
Chemical Name:	1-(4-(4-Chlorobenzyl)-4H-thieno[3,2-b]pyrrole-5-carbonyl)-N-isopropylpiperidine-4-carboxamide
Synonyms:	NCGC00112955
SMILES:	O=C(C1CCN(C(C2=CC3=C(C=CS3)N2CC4=CC=C(Cl)C=C4)=O)CC1)NC(C)C
Formula:	C₂₃H₂₆ClN₃O₂S
M.Wt:	443.99
Purity:	>98%
Sotrage:	0°C (short term), -20°C (long term), desiccated

Cat. No.	Product name	Field of application
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DC75816	Nisoxetine	Nisoxetine acts as a highly selective and potent noradrenaline transporter (NET) antagonist, exhibiting a binding affinity (Kd) of 0.76 nM. In addition to its antidepressant properties, nisoxetine functions as a local anesthetic by inhibiting voltage-gated sodium channels. This dual pharmacological activity makes it a compound of interest for both neurological and pain management research.
DC75641	GENZ-644282 TFA salt	Genz-644282, also known as SAR402674, is a non-camptothecin inhibitor of topoisomerase I with potential antineoplastic activity. Topoisomerase I inhibitor Genz-644282 binds to and inhibits the enzyme topoisomerase I, which may result in the inhibition of repair of single-strand DNA breaks, DNA replication, and tumor cell growth in susceptible tumor cell populations.
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DC74748	O4I4	O4I4 (compound 23) is a OCT4-inducing compound with metabolical stability.
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