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OS-3-106

  Cat. No.:  DC43080   Featured
Chemical Structure
1580000-17-4
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More than 5000 active chemicals with high quality for research!
Field of application
OS-3-106 represents a blood-brain barrier permeable compound demonstrating exceptional selectivity and potency as a dopamine D3 receptor (D3R) agonist. With an impressive binding affinity of Ki = 0.2 nM for D3R, this compound shows particular promise for investigating potential therapeutic interventions in psychoactive substance addiction disorders. Its unique pharmacological profile makes it a valuable research tool for studying reward system modulation.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 1580000-17-4
Chemical Name: N-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-4-(thiazol-4-yl)benzamide
Synonyms: N-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-4-(thiazol-4-yl)benzamide
SMILES: COC1C=CC=CC=1N1CCN(CCCCNC(=O)C2C=CC(C3N=CSC=3)=CC=2)CC1
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
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MSDS_26706_DC43080_1580000-17-4
COA
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Cat. No. Product name Field of application
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DC75641 GENZ-644282 TFA salt Genz-644282, also known as SAR402674, is a non-camptothecin inhibitor of topoisomerase I with potential antineoplastic activity. Topoisomerase I inhibitor Genz-644282 binds to and inhibits the enzyme topoisomerase I, which may result in the inhibition of repair of single-strand DNA breaks, DNA replication, and tumor cell growth in susceptible tumor cell populations.
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