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Home > Molecular Glues

PROTAC(H-PGDS)-7

  Cat. No.:  DC49208   Featured
Chemical Structure
2761281-50-7
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More than 5000 active chemicals with high quality for research!
Field of application
PROTAC(H-PGDS)-7 represents a breakthrough in targeted protein degradation, achieving ​unprecedented picomolar efficacy (DC50 = 17.3 pM) against hematopoietic prostaglandin D synthase (H-PGDS).
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 2761281-50-7
Chemical Name: PROTAC(H-PGDS)-7
Synonyms: 5-Pyrimidinecarboxamide, N-[4-[4-[[4-[2-(2,6-dioxo-3-piperidinyl)-2,3-dihydro-1,3-dioxo-1H-isoindol-4-yl]-1-piperazinyl]carbonyl]-1-piperidinyl]phenyl]-2-phenoxy-;PROTAC(H-PGDS)-7;2761281-50-7;CS-0311321;HY-139972;CHEMBL5076100;N-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperazine-1-carbonyl]piperidin-1-yl]phenyl]-2-phenoxypyrimidine-5-carboxamide;MS-31295;BDBM50587270
SMILES: C1(OC2=CC=CC=C2)=NC=C(C(NC2=CC=C(N3CCC(C(N4CCN(C5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)=O)CC3)C=C2)=O)C=N1
Formula: C40H38N8O7
M.Wt: 742.779128551483
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
Cat. No. Product name Field of application
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