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RY785

  Cat. No.:  DC42991   Featured
Chemical Structure
1393748-80-5
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More than 5000 active chemicals with high quality for research!
Field of application
RY785 is a potent and selective voltage-gated potassium (KV2) channel inhibitor with an IC50 of 0.05 μM for KV2.2. RY785 has analgesic activity[1].
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 1393748-80-5
Chemical Name: 3-(3-Methoxyphenyl)-2-methyl-N-[2-(1,3-thiazol-4-yl)-3H-benzimidazol-5-yl]propanamide
Synonyms: 3-(3-Methoxyphenyl)-2-methyl-n-(2-(thiazol-4-yl)-1h-benzo[d]imidazol-5-yl)propanamide;3-(3-methoxyphenyl)-2-methyl-N-(2-(thiazol-4-yl)-1H-benzo[d]imidazol-5-yl)propanamide hydrochloride;3-(3-Methoxyphenyl)-2-methyl-N-[2-(1,3-thiazol-4-yl)-3H-benzimidazol-5-yl]propanamide
SMILES: S1C=NC(=C1)C1=NC2C=CC(=CC=2N1)NC(C(C)CC1C=CC=C(C=1)OC)=O
Formula: C21H20N4O2S
M.Wt: 392.474102973938
Purity: >98%
Sotrage: 0°C (short term), -20°C (long term), desiccated
Description: RY785 is a potent and selective voltage-gated potassium (KV2) channel inhibitor with an IC50 of 0.05 μM for KV2.2. RY785 has analgesic activity[1].
Target: voltage-gated potassium (KV2) channel[1]
References: [1]. Herrington J, et al. Identification of novel and selective Kv2 channel inhibitors. Mol Pharmacol. 2011 Dec;80(6):959-64.
MSDS
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